Asst. Prof. Hacer KARATAŞ BRISTOW

Publication Network

Journal articles indexed in SCI, SSCI, and AHCI

Synthesis and Anticancer Activity of Novel Indole Derivatives as Dual EGFR/SRC Kinase Inhibitors.

Olgen S., Biltekin Kaleli S. N., Karaca B. T., Demirel U. U., Bristow H.

Current medicinal chemistry , 2023 (SCI-Expanded)

An economical and practical procedure of favipiravir synthesis for the treatment of Covid-19

Karatas H., Hanashalshahaby E. H. A., Catal U., Butun Y. E., Kurt E., Gursel S., et al.

Chemical Papers , vol.77, no.3, pp.1695-1702, 2023 (SCI-Expanded)

The Pseudo-Natural Product Rhonin Targets RHOGDI

Akbarzadeh M., Flegel J., Patil S., Shang E., Narayan R., Buchholzer M., et al.

Angewandte Chemie - International Edition , vol.61, no.18, 2022 (SCI-Expanded)

A protein tertiary structure mimetic modulator of the Hippo signalling pathway

Adihou H., Gopalakrishnan R., Förster T., Guéret S. M., Gasper R., Geschwindner S., et al.

Nature Communications , vol.11, no.1, 2020 (SCI-Expanded)

TEAD–YAP Interaction Inhibitors and MDM2 Binders from DNA-Encoded Indole-Focused Ugi Peptidomimetics

Kunig V. B. K., Potowski M., Akbarzadeh M., Klika Škopić M., dos Santos Smith D., Arendt L., et al.

Angewandte Chemie - International Edition , vol.59, no.46, pp.20338-20342, 2020 (SCI-Expanded)

Discovery of Covalent Inhibitors Targeting the Transcriptional Enhanced Associate Domain Central Pocket

KARATAŞ BRISTOW H., Akbarzadeh M., Adihou H., Hahne G., Pobbati A. V., Yihui Ng E., et al.

Journal of Medicinal Chemistry , vol.63, no.20, pp.11972-11989, 2020 (SCI-Expanded)

Identification of Quinolinols as Activators of TEAD-Dependent Transcription

Pobbati A. V., Mejuch T., Chakraborty S., KARATAŞ BRISTOW H., Bharath S. R., Guéret S. M., et al.

ACS Chemical Biology , vol.14, no.12, pp.2909-2921, 2019 (SCI-Expanded)

Real-Time Imaging and Quantification of Peptide Uptake in Vitro and in Vivo

KARATAŞ BRISTOW H., Maric T., D'Alessandro P. L., Yevtodiyenko A., Vorherr T., Hollingworth G. J., et al.

ACS Chemical Biology , vol.14, no.10, pp.2197-2205, 2019 (SCI-Expanded)

The cholesterol transfer protein GRAMD1A regulates autophagosome biogenesis

Laraia L., Friese A., Corkery D. P., Konstantinidis G., Erwin N., Hofer W., et al.

Nature Chemical Biology , vol.15, no.7, pp.710-720, 2019 (SCI-Expanded)

Chemical suppression of specific C-C chemokine signaling pathways enhances cardiac reprogramming

Guo Y., Lei I., Tian S., Gao W., Hacer K., Li Y., et al.

Journal of Biological Chemistry , vol.294, no.23, pp.9134-9146, 2019 (SCI-Expanded)

In Vivo Molecular Bioluminescence Imaging: New Tools and Applications

Mezzanotte L., van ‘t Root M., KARATAŞ BRISTOW H., Goun E. A., Löwik C. W.

Trends in Biotechnology , vol.35, no.7, pp.640-652, 2017 (SCI-Expanded)

Discovery of a Highly Potent, Cell-Permeable Macrocyclic Peptidomimetic (MM-589) Targeting the WD Repeat Domain 5 Protein (WDR5)-Mixed Lineage Leukemia (MLL) Protein-Protein Interaction

KARATAŞ BRISTOW H., Li Y., Liu L., Ji J., Lee S., Chen Y., et al.

Journal of Medicinal Chemistry , vol.60, no.12, pp.4818-4839, 2017 (SCI-Expanded)

MLL1 Inhibition Reprograms Epiblast Stem Cells to Naive Pluripotency

Zhang H., Gayen S., Xiong J., Zhou B., Shanmugam A. K., Sun Y., et al.

Cell Stem Cell , vol.18, no.4, pp.481-494, 2016 (SCI-Expanded)

Targeting MLL1 H3K4 Methyltransferase Activity in Mixed-Lineage Leukemia

Cao F., Townsend E. C., KARATAŞ BRISTOW H., Xu J., Li L., Lee S., et al.

Molecular Cell , vol.53, no.2, pp.247-261, 2014 (SCI-Expanded)

Structure-based design of high-affinity macrocyclic peptidomimetics to block the menin-mixed lineage leukemia 1 (MLL1) protein-protein interaction

Zhou H., Liu L., Huang J., Bernard D., KARATAŞ BRISTOW H., Navarro A., et al.

Journal of Medicinal Chemistry , vol.56, no.3, pp.1113-1123, 2013 (SCI-Expanded)

High-affinity, small-molecule peptidomimetic inhibitors of mll1/wdr5 protein-protein interaction

KARATAŞ BRISTOW H., Townsend E. C., Cao F., Chen Y., Bernard D., Liu L., et al.

Journal of the American Chemical Society , vol.135, no.2, pp.669-682, 2013 (SCI-Expanded)

Synthesis and potent antimicrobial activity of some novel 4-(5,6-dichloro-7H-benzimidazol-2-yl)-N-substituted benzamides

ÖZDEN M. S., KARATAŞ BRISTOW H., YILDIZ S., GÖKER A. H.

Archiv der Pharmazie , vol.337, no.10, pp.556-562, 2004 (SCI-Expanded)

Articles Published in Other Journals

Targeting Mll1 H3K4 methyltransferase activity to guide cardiac lineage specific reprogramming of fibroblasts

Liu L., Lei I., KARATAŞ BRISTOW H., Li Y., Wang L., Gnatovskiy L., et al.

Cell Discovery , vol.2, 2016 (Scopus)

MLL1 and MLL1 fusion proteins have distinct functions in regulating leukemic transcription program

Xu J., Li L., Xiong J., DenDekker A., Ye A., KARATAŞ BRISTOW H., et al.

Cell Discovery , vol.2, 2016 (Scopus)

Publications & Works